Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM269730((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
EC50: 60nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
EC50: 1.10nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
EC50: 1.10nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
EC50: 3.80nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
EC50: 60nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM269731((1R,2S)-1-(4-cyanophenyl)-N-(4-(2,6-dimethoxypheny...)
EC50: 60nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair