Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM269929((3R,5S)—N-(4-(2,6-dimethoxyphenyl)-5-(6-methy...)
BDBM269930((3R,5S)—N-(4-(2,6-dimethoxyphenyl)-5-(6-methy...)EC50: 47nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM269930((3R,5S)—N-(4-(2,6-dimethoxyphenyl)-5-(6-methy...)
BDBM363736(US9845310, Example 462.0)EC50: 9nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM269930((3R,5S)—N-(4-(2,6-dimethoxyphenyl)-5-(6-methy...)
EC50: 47nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM269930((3R,5S)—N-(4-(2,6-dimethoxyphenyl)-5-(6-methy...)
EC50: 7.80nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair