Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM269932((3R,5S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
BDBM269934((3R,5S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
EC50: 35nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair
BDBM269932((3R,5S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
BDBM269932((3R,5S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
EC50: 1.40nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM269932((3R,5S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
EC50: 35nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV-3 expression vector (Sig...More data for this Ligand-Target Pair
BDBM269935((3R,5S)N-(4-(2,6-dimethoxyphenyl)-5-(5-methy...)
EC50: 1nMpH: 7.5Assay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV¿-3 expression vector (Si...More data for this Ligand-Target Pair