Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50416858(CHEMBL1254743)Copy SMILESCopy InChI

Affinity DataKi:  0.513nMAssay Description:Displacement of [3H]prazosin from human adrenergic Alpha-1D expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
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TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50416858(CHEMBL1254743)Copy SMILESCopy InChI

Affinity DataKi:  1.12nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50416858(CHEMBL1254743)Copy SMILESCopy InChI

Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]prazosin from human adrenergic Alpha-1B expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50416858(CHEMBL1254743)Copy SMILESCopy InChI

Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]8-OH-DPAT from human adrenergic 5HT1A expressed in human HeLa cells cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI