Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034343((3aS,9aS)-1-Cyclopropylmethyl-5-methoxy-2,3,3a,4,9...)
Affinity DataKi:  721nMAssay Description:Tested for activity against 5-hydroxytryptamine 1A receptor from bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Arris Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50034343((3aS,9aS)-1-Cyclopropylmethyl-5-methoxy-2,3,3a,4,9...)
Affinity DataKi:  721nMAssay Description:Binding affinity against [3H]8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor sites in bovine hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Upjohn Laboratories

Curated by ChEMBL
LigandPNGBDBM50034343((3aS,9aS)-1-Cyclopropylmethyl-5-methoxy-2,3,3a,4,9...)
Affinity DataKi:  748nMAssay Description:Binding affinity for [3H]raclopride-labeled dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed