Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelatonin receptor type 1A/1B/1C(Gallus gallus)
University Of Groningen

Curated by ChEMBL

LigandBDBM50231297(CHEMBL99778)Copy SMILESCopy InChI

Affinity DataKi:  2.31E+4nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL

LigandBDBM50231297(CHEMBL99778)Copy SMILESCopy InChI

Affinity DataIC50:  22nMAssay Description:Inhibition of 2-[125I]iodomelatonin stimulated calcium dependent dopamine release from the rabbit retina.More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI