Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144161(CHEMBL65021 | N-(1-Methoxy-6-phenyl-6H-benzo[c]chr...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]dexamethasone from human Glucocorticoid receptor (GR); Value ranges from 17-21 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144161(CHEMBL65021 | N-(1-Methoxy-6-phenyl-6H-benzo[c]chr...)
Affinity DataIC50:  87nMAssay Description:Effect on human Glucocorticoid receptor (GR) in a whole cell assay to measure functional cellular GR-antagonism (GRAF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144161(CHEMBL65021 | N-(1-Methoxy-6-phenyl-6H-benzo[c]chr...)
Affinity DataIC50:  3.36E+3nMAssay Description:Displacement of [3H]progesterone from human Progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144161(CHEMBL65021 | N-(1-Methoxy-6-phenyl-6H-benzo[c]chr...)
Affinity DataIC50:  6.53E+3nMAssay Description:Displacement of [3H]mibolerone from human Androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144161(CHEMBL65021 | N-(1-Methoxy-6-phenyl-6H-benzo[c]chr...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]estradiol from human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144161(CHEMBL65021 | N-(1-Methoxy-6-phenyl-6H-benzo[c]chr...)
Affinity DataIC50:  2.29E+4nMAssay Description:Displacement of [3H]aldosterone from human Mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed