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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Melanocyte-stimulating hormone receptor
(Mus musculus)
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217722
((2R,E)-2-amino-N-(4-ethyl-4-(methylamino)octyl)-3-...)
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Affinity Data
Ki: 1.60E+3nM
Assay Description:
Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Melanocortin receptor 4
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217722
((2R,E)-2-amino-N-(4-ethyl-4-(methylamino)octyl)-3-...)
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Affinity Data
Ki: 4.10E+3nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC4 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217722
((2R,E)-2-amino-N-(4-ethyl-4-(methylamino)octyl)-3-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4.10E+3nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC4 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217722
((2R,E)-2-amino-N-(4-ethyl-4-(methylamino)octyl)-3-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5.00E+3nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC5 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217722
((2R,E)-2-amino-N-(4-ethyl-4-(methylamino)octyl)-3-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 5.00E+3nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC5 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217722
((2R,E)-2-amino-N-(4-ethyl-4-(methylamino)octyl)-3-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.10E+4nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC3 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI