Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Siena Biotech

Curated by ChEMBL

LigandBDBM50319675(1-(2'-methoxybiphenyl-4-yl)-3-(4-(piperidin-1-yl)b...)Copy SMILESCopy InChI

Affinity DataIC50:  7.80E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Siena Biotech

Curated by ChEMBL

LigandBDBM50319675(1-(2'-methoxybiphenyl-4-yl)-3-(4-(piperidin-1-yl)b...)Copy SMILESCopy InChI

Affinity DataEC50:  140nMAssay Description:Displacement of [3H]epibatidine from rat alpha7 nAChR expressed in rat GH4C1 cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI