Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50416773(CHEMBL1242352)
Affinity DataKi:  0.263nMAssay Description:Displacement [3H]prazosin of human recombinant alpha1A adrenergic receptor expressed in CHO cells by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50416773(CHEMBL1242352)
Affinity DataKi:  0.813nMAssay Description:Displacement [3H]prazosin of human recombinant Alpha-1D adrenergic receptor expressed in CHO cells by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50416773(CHEMBL1242352)
Affinity DataKi:  6.76nMAssay Description:Displacement [3H]prazosin of human recombinant Alpha-1B adrenergic receptor expressed in CHO cells by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50416773(CHEMBL1242352)
Affinity DataKi:  15.1nMAssay Description:Binding affinity to 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50416773(CHEMBL1242352)
Affinity DataKi:  22.9nMAssay Description:Displacement [3H]8-OH-DPAT of human cloned 5HT1A receptor expressed in human HeLa cells by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed