Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Vu University Medical Center

Curated by ChEMBL
LigandPNGBDBM50343889(3-Iodo-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)eth...)
Affinity DataKi:  2.15nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptor expressed in HEK293 EBNA cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Vu University Medical Center

Curated by ChEMBL
LigandPNGBDBM50343889(3-Iodo-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)eth...)
Affinity DataIC50:  5.04nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptor expressed in HEK293 EBNA cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed