Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  960nMAssay Description:Inhibition of VEGFR2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of Src by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of TIE2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of IGF1R by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of EGFR by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of VEGFR3 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora B by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of insulin receptor by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Aurora A by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50248182(CHEMBL475351 | N-(4-(benzo[d]thiazol-2-yl)-3-metho...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ErbB2 by virtual HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed