Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL

LigandBDBM50108095(CHEMBL3601310)Copy SMILESCopy InChI

Affinity DataEC50:  111nMAssay Description:Agonist activity at human recombinant beta3-adrenergic receptor expressed in CHO cells assessed as increase of cAMP level after 30 minsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Asahi Kasei Pharma

Curated by ChEMBL

LigandBDBM50108095(CHEMBL3601310)Copy SMILESCopy InChI

Affinity DataEC50:  33nMAssay Description:Agonist activity at human alpha1A-adrenergic receptor expressed in HEK293 cells assessed as calcium flux by fluorescence assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI