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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Leucine-rich repeat serine/threonine-protein kinase 2
(Homo sapiens (Human))
Imago Pharmaceuticals
US Patent
Ligand
BDBM50428710
(CHEMBL2333134 | US9884828, 2-23)
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Affinity Data
IC50: 17nM
pH: 7.5 T: 2°C
Assay Description:
Compounds as described herein (compounds of Formula I, e.g., compounds of the above Examples) are tested for their in vitro kinase activities using v...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
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Target
Leucine-rich repeat serine/threonine-protein kinase 2
(Homo sapiens (Human))
Imago Pharmaceuticals
US Patent
Ligand
BDBM50428710
(CHEMBL2333134 | US9884828, 2-23)
Copy SMILES
Copy InChI
Affinity Data
IC50: 17nM
Assay Description:
Inhibition of wild type GST-tagged LRRK2 (970 to 2527 amino acid residues) (unknown origin) assessed as inhibition of biotinylated-LRRKtide phosphory...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI