Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMetallo-beta-lactamase L1 type 3(Stenotrophomonas maltophilia)
North-West University

Curated by ChEMBL
LigandPNGBDBM50092976(CHEMBL3586478)
Affinity DataKi:  110nMAssay Description:Mixed-type inhibition of Stenotrophomonas maltophilia L1 overexpressed in Escherichia coli BL21 (DE3) using imipenem as substrate incubated for 30 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase L1 type 3(Stenotrophomonas maltophilia)
North-West University

Curated by ChEMBL
LigandPNGBDBM50092976(CHEMBL3586478)
Affinity DataIC50:  18nMAssay Description:Inhibition of Stenotrophomonas maltophilia L1 overexpressed in Escherichia coli BL21 (DE3) using imipenem as substrate incubated for 30 mins prior to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
North-West University

Curated by ChEMBL
LigandPNGBDBM50092976(CHEMBL3586478)
Affinity DataIC50:  1.23E+5nMAssay Description:Inhibition of Bacteroides fragilis CcrA overexpressed in Escherichia coli BL21 (DE3) using cefazolin as substrate incubated for 30 mins prior to test...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed