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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065057(1-(4-Fluoro-benzyl)-3-(6-methyl-2,4-bis-methylsulf...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase (ACAT) in rabbit intestinal microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50065057(1-(4-Fluoro-benzyl)-3-(6-methyl-2,4-bis-methylsulf...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity towards ACAT by the displacement of [1-14C]-oleolyl-CoA from the small intestine of cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed