Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50190268
(4'-methylsulfanyl-biphenyl-4-carboxylic acid methy...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4nM
Assay Description:
Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
Neurocrine Biosciences
Curated by
ChEMBL
Ligand
BDBM50190268
(4'-methylsulfanyl-biphenyl-4-carboxylic acid methy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.20nM
Assay Description:
Antagonist activity against human MCHR1 expressed in CHO cells assessed by inhibition of MCH-stimulated G protein-GTPgamma35S binding
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI