Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190268(4'-methylsulfanyl-biphenyl-4-carboxylic acid methy...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I-Tyr13]MCH from human MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50190268(4'-methylsulfanyl-biphenyl-4-carboxylic acid methy...)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells assessed by inhibition of MCH-stimulated G protein-GTPgamma35S bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed