Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM50080292(4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidi...)Ki: 25nMAssay Description:Inhibitory activity against binding of the [3H]-DPCPX to human A1 receptor (hA1) radioligands using competition binding assayMore data for this Ligand-Target Pair
BDBM50080292(4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidi...)
BDBM50080292(4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidi...)
BDBM50080292(4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidi...)
IC50: 49nMAssay Description:Binding affinity against human A2 receptor (hA2) was measured through displacement of [3H]-CGS-21,680 using yeast cell membranesMore data for this Ligand-Target Pair
BDBM50080292(4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidi...)
IC50: 1.54E+3nMAssay Description:Inhibitory activity against binding of [3H]-CGS-21,680 to human A2a receptor (hA2a) using competition binding assayMore data for this Ligand-Target Pair
BDBM50080292(4-(5,6-Dimethyl-2-phenyl-7H-pyrrolo[2,3-d]pyrimidi...)
IC50: 1.62E+3nMAssay Description:Binding affinity against human A1 receptor (hA1) was measured through displacement of [3H]-DPCPX using yeast cell membranesMore data for this Ligand-Target Pair