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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Apoptosis regulator Bcl-2
(Homo sapiens (Human))
Ucb Pharma
Curated by
ChEMBL
Ligand
BDBM50254584
(4-chloro-1-(2-((S)-3-(hydroxymethyl)-1,2,3,4-tetra...)
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Affinity Data
IC50: 50nM
Assay Description:
Inhibition of GST fused Bcl-2 (unknown origin) binding to biotinylated 16 mer Bak-BH3 peptide by HTRF-LANCE assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Apoptosis regulator Bcl-2
(Homo sapiens (Human))
Ucb Pharma
Curated by
ChEMBL
Ligand
BDBM50254584
(4-chloro-1-(2-((S)-3-(hydroxymethyl)-1,2,3,4-tetra...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 480nM
Assay Description:
Inhibition of GST fused Bcl-2 (unknown origin) binding to biotinylated 26 mer Bak-BH3 peptide by HTRF-LANCE assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Bcl2-associated agonist of cell death
(Homo sapiens (Human))
Ucb Pharma
Curated by
ChEMBL
Ligand
BDBM50254584
(4-chloro-1-(2-((S)-3-(hydroxymethyl)-1,2,3,4-tetra...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.28E+3nM
Assay Description:
Inhibition of GST fused Bcl-xL (unknown origin) binding to biotinylated 16 mer Bak-BH3 peptide by HTRF-LANCE assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI