Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  28nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  28nMAssay Description:Inhibition of [3H]dexamethasone binding to human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  28nMAssay Description:Inhibition of [3H]-dexamethasone binding to glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  170nMAssay Description:Displacement of [3H]-dexamethasone from human androgen receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  250nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  250nMAssay Description:Inhibition of glucocorticoid receptor Dexamethasone response in reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  250nMAssay Description:Inhibition of glucocorticoid receptor dexamethasone responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]-dexamethasone from human mineralocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144457(CHEMBL419633 | N-(3-Dibenzylamino-2-methyl-phenyl)...)
Affinity DataIC50:  7.60E+3nMAssay Description:Displacement of [3H]-dexamethasone from human progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed