Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008964(2,6-Di-tert-butyl-4-[2-(3-methyl-isoxazol-5-yl)-vi...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against cyclooxygenase in rat basophilic leukemia cells using prostaglandin G/H synthase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008964(2,6-Di-tert-butyl-4-[2-(3-methyl-isoxazol-5-yl)-vi...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity against 5-lipoxygenase in rat basophilic leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50008964(2,6-Di-tert-butyl-4-[2-(3-methyl-isoxazol-5-yl)-vi...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of 5-lipoxygenase measured by the reduction of leukotriene B4 (LTB4) in intact basophilic rat leukemia cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed