Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
B2 bradykinin receptor
(Homo sapiens (Human))
Jerini
Curated by
ChEMBL
Ligand
BDBM50293878
(4-(5-chloro-thiazol-4-yl)-8-(3,5-dichloro-pyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 210nM
Assay Description:
Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
B2 bradykinin receptor
(Homo sapiens (Human))
Jerini
Curated by
ChEMBL
Ligand
BDBM50293878
(4-(5-chloro-thiazol-4-yl)-8-(3,5-dichloro-pyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 730nM
Assay Description:
Antagonist activity at B2 receptor in human HF15 cells assessed as inhibition of bradykinin-induced calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI