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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM48131(1H-indazole-3-carboxylic acid [2-keto-2-(1,2,5-tri...)
Affinity DataIC50:  3.24E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetMatrix metalloproteinase-14 [1-36](Homo sapiens (Human))
Sanford-Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48131(1H-indazole-3-carboxylic acid [2-keto-2-(1,2,5-tri...)
Affinity DataEC50:  7.21E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay