Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetB2 bradykinin receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50419894(CHEMBL1956871)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50419894(CHEMBL1956871)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H][desArg9]Lys-Bradykinin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50419894(CHEMBL1956871)
Affinity DataKd:  5.01nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed