Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
IC50: 88nMpH: 7.4Assay Description:The TACE enzyme is an internal production (carried out according to the publication protein Eng Des Sel, 2006, 19, 155-161) and is added so as to hav...More data for this Ligand-Target Pair
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
IC50: 2.61E+3nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
IC50: 5.80E+3nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
Stromelysin-1(Homo sapiens (Human))Galderma Research & Development
US Patent
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
IC50: 6.83E+3nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
IC50: >1.00E+4nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
BDBM175083(US9115102, Ex14 | US9115102, Ex24)
IC50: >1.00E+4nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair