Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL

LigandBDBM50204396((3S,4S)-N-hydroxy-4-(4-((2-methylquinolin-4-yl)met...)Copy SMILESCopy InChI

Affinity DataIC50: <1nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair

Target InfoPDBMMDB
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL

LigandBDBM50204396((3S,4S)-N-hydroxy-4-(4-((2-methylquinolin-4-yl)met...)Copy SMILESCopy InChI

Affinity DataIC50:  67nMAssay Description:Inhibition of TACE in human whole bloodMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI