Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 1 hits in this display
BDBM50220082(2-(3-fluoro-5-methylphenyl)pyrido[2,3-d]pyrimidine...)
IC50: 321nMAssay Description:Antagonistic activity at rat mGluR5 expressed in CHO cells assessed as inhibition of quisqualate stimulated calcium mobilization by FLIPR technologyMore data for this Ligand-Target Pair