Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataKi:  0.111nMAssay Description:Inhibition of [3H]-DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataKi:  594nMAssay Description:Inhibition of [3H]-DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataIC50:  2.31nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataIC50:  46.4nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed