Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMu-type opioid receptor(GUINEA PIG)
National University Of Singapore

Curated by ChEMBL

LigandBDBM50252864(CHEMBL454035 | antanal 2)Copy SMILESCopy InChI

Affinity DataKi:  1.52nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetDelta-type opioid receptor(MOUSE)
National University Of Singapore

Curated by ChEMBL

LigandBDBM50252864(CHEMBL454035 | antanal 2)Copy SMILESCopy InChI

Affinity DataKi:  7.74nMAssay Description:Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced responseMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI