Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 13 hits in this display
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Ki: 0.810nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranes incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Ki: 520nMAssay Description:Displacement of [3H]U-69593 from human recombinant KOR expressed in CHO cell membranes incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
IC50: 0.260nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
IC50: 0.590nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
BDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)