Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50207192
((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.600nM
Assay Description:
Displacement of [3H]DAMGO 2 from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50207192
((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1nM
Assay Description:
Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50207192
((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 553nM
Assay Description:
Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated contraction
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI