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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
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kcal/mol
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Found
1
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Target
Neuronal acetylcholine receptor subunit alpha-4
(Homo sapiens (Human))
Amgen
Curated by
ChEMBL
Ligand
BDBM50264765
(3-methyl-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)iso...)
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Affinity Data
EC50: 1.30E+3nM
Assay Description:
Activation of human alpha4beta2 nAChR assessed as potentiation of submaximal response to nicotine induced current
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