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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Neuronal acetylcholine receptor; alpha9/alpha10
(Homo sapiens (Human))
University Of Kentucky
Curated by
ChEMBL
Ligand
BDBM50339934
(1,1'-(3,3'-(biphenyl-4,4'-diyl)bis(propane-3,1-diy...)
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Affinity Data
IC50: 4.20nM
Assay Description:
Antagonist activity at alpha9/alpha10 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-gated current by voltage clamp electrophysiolog...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Neuronal acetylcholine receptor subunit alpha-7
(Homo sapiens (Human))
University Of Kentucky
Curated by
ChEMBL
Ligand
BDBM50339934
(1,1'-(3,3'-(biphenyl-4,4'-diyl)bis(propane-3,1-diy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.51E+3nM
Assay Description:
Antagonist activity at alpha7 nAChR expressed in Xenopus oocyte assessed as inhibition of ACh-gated current by voltage clamp electrophysiology assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI