Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50377935(CHEMBL541164)
Affinity DataKi:  2.97E+4nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50377935(CHEMBL541164)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50377935(CHEMBL541164)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed