Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetD(4) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by ChEMBL
LigandPNGBDBM50124936(2,2-Dimethyl-5-[4-(4-methyl-benzyl)-piperazin-1-yl...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-YM 09151 from D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Neurogen

Curated by ChEMBL
LigandPNGBDBM50124936(2,2-Dimethyl-5-[4-(4-methyl-benzyl)-piperazin-1-yl...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]-YM 09151 from D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Neurogen

Curated by ChEMBL
LigandPNGBDBM50124936(2,2-Dimethyl-5-[4-(4-methyl-benzyl)-piperazin-1-yl...)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]prazosin from alpha-1 adrenergic receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed