Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Wyeth-Ayerst Research

Curated by ChEMBL

LigandBDBM50078663(CHEMBL300946 | N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a]...)Copy SMILESCopy InChI

Affinity DataIC50:  4nMAssay Description:In vitro inhibition of (P[3H]-AVP binding to isolated rat kidney medullary V2 receptorMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetVasopressin V1a receptor(RAT)
Wyeth-Ayerst Research

Curated by ChEMBL

LigandBDBM50078663(CHEMBL300946 | N-[5-(5H,11H-Benzo[e]pyrrolo[1,2-a]...)Copy SMILESCopy InChI

Affinity DataIC50:  33nMAssay Description:Displacement of (Phe-3,4,5 [3H]-) AVP from isolated rat hepatic V1a receptorMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI