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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341235(4-(aminomethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)pyr...)
Affinity DataIC50:  788nMAssay Description:Inhibition of human wild type KIT assessed as [gamma33P]ATP incorporation into polyGluTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341235(4-(aminomethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)pyr...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of human wild type PDGFRalpha assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50341235(4-(aminomethyl)-N-(4-methyl-3-(4-(pyridin-3-yl)pyr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human wild type ABL1 assessed as [gamma33P]ATP incorporation into polyAlaGluLsTyr after 60 mins by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed