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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50:  5.70nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50:  6.30nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50:  6.60nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: <10nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: <13nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50:  140nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 6(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
University Of Washington

LigandPNGBDBM81376(Amine compound, 13a)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed