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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50154998
(2-[2-(5-Fluoro-4''-methyl-biphenyl-3-yl)-2H-tetraz...)
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Affinity Data
IC50: 1.47E+3nM
Assay Description:
In vitro antagonistic activity against Metabotropic glutamate receptor 5 in [Ca2+] flux assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50154998
(2-[2-(5-Fluoro-4''-methyl-biphenyl-3-yl)-2H-tetraz...)
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Copy InChI
Affinity Data
IC50: >3.00E+3nM
Assay Description:
Antagonistic activity of the compound against Metabotropic glutamate receptor 5 in [Ca2+] flux assay using glutamate (10 uM) as agonist
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI