Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL

LigandBDBM50362362(CHEMBL1939759)Copy SMILESCopy InChI

Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]-DAK from human bradykinin B1 receptor expressed in CHO-D-/aequorin cells membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL

LigandBDBM50362362(CHEMBL1939759)Copy SMILESCopy InChI

Affinity DataIC50:  0.230nMAssay Description:Antagonist activity at human bradykinin B1 receptor expressed in CHO-D-/aequorin cells assessed as inhibition of DAK-induced intracellular calcium le...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI