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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Vanderbilt University School Of Medicine
Curated by
ChEMBL
Ligand
BDBM50187633
(3,4-dimethyl-N-(1,3-diphenyl-1H-pyrazol-5-yl)benza...)
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Affinity Data
Ki: 430nM
Assay Description:
Displacement of [3H]methoxyPEPy from rat mGluR5 expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Vanderbilt University School Of Medicine
Curated by
ChEMBL
Ligand
BDBM50187633
(3,4-dimethyl-N-(1,3-diphenyl-1H-pyrazol-5-yl)benza...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 20nM
Assay Description:
Activity at mGluR5 assessed as potentiation of glutamate-induced calcium flux in rat astrocytes
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI