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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [3H]mesulergine at human cloned 5HT2C receptor expressed in CHOK1 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from human cloned 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]8-OH-DPAT from human cloned 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Korea Research Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50251611(5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed