Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCarbonic anhydrase(Candida glabrata)
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50158512(CHEMBL3787222)
Affinity DataKi:  30nMAssay Description:Inhibition of recombinant Candida glabrata beta carbonic anhydrase NCE103 expressed in Escherichia coli preincubated for 15 mins by stopped-flow CO2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Candida albicans (Yeast))
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50158512(CHEMBL3787222)
Affinity DataKi:  128nMAssay Description:Inhibition of recombinant Candida albicans beta carbonic anhydrase NCE103 expressed in Escherichia coli preincubated for 15 mins by stopped-flow CO2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50158512(CHEMBL3787222)
Affinity DataKi:  414nMAssay Description:Inhibition of recombinant human carbonic anhydrase 1 expressed in Escherichia coli preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Bezmialem Vakif University

Curated by ChEMBL
LigandPNGBDBM50158512(CHEMBL3787222)
Affinity DataKi:  454nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 expressed in Escherichia coli preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed