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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 14 hits in this display   

TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataIC50:  169nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataIC50:  169nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  33nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  97nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  678nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  33nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse BRS3 expressed in HEK293 cells expressing aequorin measured for 30 secs by bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  677nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human BRS3 expressed in HEK293 cells expressing aequorin measured for 10 mins by bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in HEK293 cells expressing aequorin measured for 30 secs by bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  97nMAssay Description:Agonist activity at human BRS3 expressed in HEK293 cells expressing aequorin measured for 30 secs by bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  97nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  33nMAssay Description:Agonist activity at mouse BRS3 expressed in HEK293 cells expressing aequorin measured for 30 secs by bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed