Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50171759(7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-ca...)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to adenosine A2a receptor of human striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50171759(7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-ca...)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]-CGS-21,680 binding to adenosine A2a receptor of bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50171759(7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-ca...)
Affinity DataKi:  300nMAssay Description:Inhibition of [3H]-CHA binding to adenosine A1 receptor of human brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Dipartimento Di Scienze Farmaceutiche

Curated by ChEMBL
LigandPNGBDBM50171759(7-Methyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-ca...)
Affinity DataKi:  1.35E+3nMAssay Description:Inhibition of [3H]-CHA binding to adenosine A1 receptor of bovine brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed