Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  151nMAssay Description:Binding affinity to human alpha1B adrenergic receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]-prazosin from human alpha1B adrenergic receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  479nMAssay Description:Displacement of [3H]-prazosin from human alpha1D adrenergic receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  479nMAssay Description:Binding affinity to human alpha1D adrenergic receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  617nMAssay Description:Binding affinity to human alpha1A adrenergic receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  617nMAssay Description:Displacement of [3H]-prazosin from human alpha1A adrenergic receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human 5HT1A receptor transfected in COS1 cells assessed as compound required to occupy 50% of receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Unsw Australia

Curated by ChEMBL
LigandPNGBDBM50103891(CHEMBL3343980)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor transfected in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed