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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Kobe Gakuin University
Curated by
ChEMBL
Ligand
BDBM50212613
(CHEMBL266122 | Tyr-Pro-Dmp-Phe-NH2)
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Affinity Data
Ki: 0.0440nM
Assay Description:
Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Kobe Gakuin University
Curated by
ChEMBL
Ligand
BDBM50212613
(CHEMBL266122 | Tyr-Pro-Dmp-Phe-NH2)
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Copy InChI
Affinity Data
Ki: 1.44E+3nM
Assay Description:
Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Kobe Gakuin University
Curated by
ChEMBL
Ligand
BDBM50212613
(CHEMBL266122 | Tyr-Pro-Dmp-Phe-NH2)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Displacement of [3H]U69,593 from kappa opioid receptor in Hartley guinea pig cerebellum P2 synaptosome membrane
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
Kobe Gakuin University
Curated by
ChEMBL
Ligand
BDBM50212613
(CHEMBL266122 | Tyr-Pro-Dmp-Phe-NH2)
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Affinity Data
IC50: 0.380nM
Assay Description:
Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contraction
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(MOUSE)
Kobe Gakuin University
Curated by
ChEMBL
Ligand
BDBM50212613
(CHEMBL266122 | Tyr-Pro-Dmp-Phe-NH2)
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Affinity Data
IC50: 1.39nM
Assay Description:
Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI