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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM50201484
(CHEMBL396691 | N-(6-methylpyridin-2-yl)-2-oxo-2,3-...)
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Affinity Data
Ki: 95nM
Assay Description:
Binding affinity to mGluR5
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by
ChEMBL
Ligand
BDBM50201484
(CHEMBL396691 | N-(6-methylpyridin-2-yl)-2-oxo-2,3-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 60nM
Assay Description:
Antagonist activity at mGluR5 assessed as inhibition of Ca2+ efflux by FLIPR
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI