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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCarbonic anhydrase 1(Homo sapiens (Human))
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258715(1-({[5-(Aminosulfonyl)-3-(3-bromophenyl)-1H-indol-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human recombinant CA1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258715(1-({[5-(Aminosulfonyl)-3-(3-bromophenyl)-1H-indol-...)
Affinity DataKi:  7.80nMAssay Description:Inhibition of human recombinant CA2 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Candida albicans (Yeast))
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258715(1-({[5-(Aminosulfonyl)-3-(3-bromophenyl)-1H-indol-...)
Affinity DataKi:  64nMAssay Description:inhibition of Candida albicans recombinant Nce103 after 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase(Mycobacterium tuberculosis)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258715(1-({[5-(Aminosulfonyl)-3-(3-bromophenyl)-1H-indol-...)
Affinity DataKi:  104nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant carbonic anhydrase Rv3273 by by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-carbonic anhydrase 1(Mycobacterium tuberculosis)
Istanbul University

Curated by ChEMBL
LigandPNGBDBM50258715(1-({[5-(Aminosulfonyl)-3-(3-bromophenyl)-1H-indol-...)
Affinity DataKi:  110nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant carbonic anhydrase Rv1284 by by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed