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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant GST-fused ALK5 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  540nMAssay Description:Inhibition of p38alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  650nMAssay Description:Inhibition of PKCmuMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  940nMAssay Description:Inhibition of VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of VEGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50320964(3-((4-(6-Methylpyridin-2-yl)-5-(quinolin-6-yl)-1H-...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed